What is the mechanism of action of Tapentadol 100mg?

What is the mechanism of action of Tapentadol 100mg?

What is Tapentadol?

Tapentadol is a prescription medication belonging to the class of opioid analgesics. It works by binding to the opioid receptors in the brain and spinal cord, reducing the sensation of pain.

How does Tapentadol work?

Tapentadol blocks the reuptake of neurotransmitters norepinephrine and serotonin in the brain. By increasing their concentration, it reduces the perception of pain. Additionally, tapentadol binds to mu-opioid receptors, further reducing pain perception.

The Dual Mechanism of Action

Unlike other opioids, tapentadol has a dual mechanism of action. It effectively relieves chronic pain, neuropathic pain, and acute pain caused by injury or surgery.

Important Considerations

It is crucial to note that tapentadol can be habit-forming and lead to dependence if used for a prolonged period. Only take tapentadol as prescribed by a healthcare professional and follow the recommended dosing schedule. Abruptly stopping the medication can result in severe withdrawal symptoms.


Tapentadol is an effective pain reliever that works by blocking neurotransmitter reuptake and activating mu-opioid receptors. To avoid dependence and withdrawal symptoms, it is essential to use this medication as prescribed. If you have any questions or concerns about tapentadol or its use, consult your healthcare provider. To buy Tapentadol online, visit our website today.

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